Tivantinib for second-line treatment of advanced hepatocellular carcinoma: a randomised, placebo-controlled phase 2 study

Armando Santoro, Lorenza Rimassa, Ivan Borbath, Bruno Daniele, Stefania Salvagni, Jean Luc Van Laethem, Hans Van Vlierberghe, Jörg Trojan, Frank T Kolligs, Alan Weiss, Steven Miles, Antonio Gasbarrini, Monica Lencioni, Luca Cicalese, Morris Sherman, Cesare Gridelli, Peter Buggisch, Guido Gerken, Roland M Schmid, Corrado BoniNicola Personeni, Ziad Hassoun, Giovanni Abbadessa, Brian Schwartz, Reinhard Von Roemeling, Maria E Lamar, Yinpu Chen, Camillo Porta

Risultato della ricerca: Contributo in rivistaArticolo in rivista

436 Citazioni (Scopus)

Abstract

Tivantinib (ARQ 197), a selective oral inhibitor of MET, has shown promising antitumour activity in hepatocellular carcinoma as monotherapy and in combination with sorafenib. We aimed to assess efficacy and safety of tivantinib for second-line treatment of advanced hepatocellular carcinoma.
Lingua originaleEnglish
pagine (da-a)55-63
Numero di pagine9
RivistaThe Lancet Oncology
Volume14
DOI
Stato di pubblicazionePubblicato - 2013

Keywords

  • Adult
  • Aged
  • Aged, 80 and over
  • Carcinoma, Hepatocellular
  • Disease-Free Survival
  • Double-Blind Method
  • Drug-Related Side Effects and Adverse Reactions
  • Female
  • Gene Expression
  • Humans
  • Kaplan-Meier Estimate
  • Liver Neoplasms
  • Male
  • Middle Aged
  • Neoplasm Staging
  • Protein Kinase Inhibitors
  • Proto-Oncogene Proteins c-met
  • Pyrrolidinones
  • Quinolines

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